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membrane MDR1 ABCB1
membrane transporter MDR1 ABCB1
MDR1 assay
transporter MDR1 ABCB1
P-glycoprotein MDR1 ABCB1
multidrug resistance MDR1 ABCB1
chemotheraphy MDR1 ABCB1
blood-brain barrier MDR2 ABCB2
BBB MDR1 ABCB1
assay MDR1 ABCB1
transport MDR1 ABCB1
screening MDR1 ABCB1
ADME MDR1 ABCB1
Absorption MDR1 ABCB1
Distribution MDR1 ABCB1
Metabolism MDR1 ABCB1
Excretion MDR1 ABCB1
early ADME MDR1 ABCB1
in-vitro system MDR1 ABCB1
drug metabolism MDR1 ABCB1
nucleotide trapping MDR1 ABCB1
dye transport MDR1 ABCB1
bioavailability MDR1 ABCB1
xenobiotics MDR1 ABCB1
permeability MDR1 ABCB1
cancer drug resistance MDR1 ABCB1
hydrophobic drug MDR1 ABCB1
drug interaction MDR1 ABCB1
modulator MDR1 ABCB1
pharmacokinetics MDR1 ABCB1
CNS penetration MDR1 ABCB1
modulator MDR1 ABCB1
Ivermectin MDR1 ABCB1
DMPK MDR1 ABCB1
chemotherapy MDR1 ABCB1
resistant tumor cell MDR1 ABCB1
anticancer drug MDR1 ABCB1
chemosensitizer MDR1 ABCB1
lead optimization MDR1 ABCB1
drug development MDR2 ABCB2
HTS MDR1 ABCB1
pharmacology MDR1 ABCB1
Paclitaxel MDR1 ABCB1
PSC833 MDR1 ABCB1
cyclosporin A MDR1 ABCB1
somatostatin MDR1 ABCB1
somatostatin analogues MDR2 ABCB2
Ivermectin MDR1 ABCB1
indinavir MDR1 ABCB1
deaxamethasone MDR1 ABCB1
digoxin MDR1 ABCB1
doxorubicin MDR1 ABCB1
vecuronium MDR1 ABCB1
azido-procainamide MDR1 ABCB1
tributyltrimethylammonium MDR1 ABCB1
rifampin MDR1 ABCB1
tacrolimus MDR1 ABCB1
vinblastine MDR1 ABCB1
ondansteron MDR1 ABCB1
quinidine MDR1 ABCB1
verapamil MDR1 ABCB1
loperamide MDR1 ABCB1
CsA MDR1 ABCB1
GG918 MDR1 ABCB1
talinolol MDR1 ABCB1
fexofenidine MDR1 ABCB1
fexofenadine MDR2 ABCB2
actinomycin D MDR1 ABCB1
Vinca alkaloides MDR1 ABCB1
taxanes MDR1 ABCB1
anthracyclines MDR1 ABCB1
epipodophyllotoxins MDR1 ABCB1
antheacenes MDR1 ABCB1
colchicine MDR1 ABCB1
saquinavir MDR1 ABCB1
ritonavir MDR1 ABCB1
amprenavir MDR1 ABCB1
nelfinavir MDR1 ABCB1
lopinavir MDR1 ABCB1
FK506 MDR1 ABCB1
erythromycin MDR1 ABCB1
domperidone MDR1 ABCB1
cimetidine MDR1 ABCB1
diltiazam MDR1 ABCB1
morphine MDR1 ABCB1
terfenidine MDR1 ABCB1
terfenadine MDR2 ABCB2
gramicidin D MDR1 ABCB1
Rhodamine123 MDR1 ABCB1
cortisol MDR1 ABCB1
loperamide MDR1 ABCB1
valinomycin MDR1 ABCB1
talinolol MDR1 ABCB1
Flavopiridol MDR1 ABCB1
Genistein MDR1 ABCB1
Isoflavone MDR1 ABCB1
Quercetin MDR1 ABCB1
amiloride MDR1 ABCB1
amiodarone MDR1 ABCB1
atorvastatin MDR1 ABCB1
Chloroquine MDR1 ABCB1
Chloropromazine MDR1 ABCB1
Clofazimine MDR1 ABCB1
cremophor EL MDR1 ABCB1
daunorubicine MDR1 ABCB1
daunomycine MDR1 ABCB1
morpholine doxorubicine MDR1 ABCB1
Diltiazem MDR1 ABCB1
Dipyridamole MDR1 ABCB1
Erythromycine MDR1 ABCB1
Fluoroquinolones MDR1 ABCB1
fleroxacin MDR1 ABCB1
enoxacin MDR1 ABCB1
grepafloxacin MDR1 ABCB1
levofloxacin MDR1 ABCB1
norfloxacine MDR1 ABCB1
Glibenclamides MDR1 ABCB1
Gramicidin MDR1 ABCB1
Hydrocortisone MDR1 ABCB1
Itraconazole MDR1 ABCB1
Lidocaine MDR1 ABCB1
propafenone MDR1 ABCB1
propanolol MDR1 ABCB1
quinine MDR1 ABCB1
quinacrine MDR1 ABCB1
cinchonine MDR1 ABCB1
SDZ PSC 833 MDR1 ABCB1
tamoxifene MDR1 ABCB1
nifedipine MDR1 ABCB1
bepridil MDR1 ABCB1
nicardipine MDR1 ABCB1
niguldipine MDR1 ABCB1
nitrendipine MDR1 ABCB1
trifluoperazine MDR1 ABCB1
felodipine MDR1 ABCB1
vincristine MDR1 ABCB1
vindesine MDR1 ABCB1
adriamycin MDR1 ABCB1
aldosteron MDR1 ABCB1
benzopyrene MDR1 ABCB1
Calcein AM MDR1 ABCB1
estradiol MDR1 ABCB1
ethidium bromide MDR1 ABCB1
etoposide MDR1 ABCB1
teniposide MDR1 ABCB1
fluo-3 MDR1 ABCB1
Hoechst 33342 MDR1 ABCB1
L-DOPA MDR1 ABCB1
Losartan MDR1 ABCB1
mithramycin MDR1 ABCB1
mitomycin C MDR1 ABCB1
docetaxel MDR1 ABCB1
puromycin MDR1 ABCB1
Tc99m sestamibi MDR1 ABCB1
topotecan MDR1 ABCB1
bergamottin MDR1 ABCB1
clarithromycin MDR1 ABCB1
dimetyl-ß-cyclodextrin MDR1 ABCB1
GF120918 MDR1 ABCB1
ketoconazole MDR1 ABCB1
LY335979 MDR1 ABCB1
midazolam MDR1 ABCB1
progesterone MDR1 ABCB1
RU 486 MDR1 ABCB1
megestrol acetate MDR1 ABCB1
testosterone MDR1 ABCB1
XR 9576 MDR1 ABCB1
XR 9051 MDR1 ABCB1
3-methyl-cholanthrene MDR1 ABCB1
phenothiazines MDR1 ABCB1
prazosin MDR1 ABCB1
prazosin MDR1 ABCB1
membrane MRP1 ABCC1
chemical toxicity MRP1 ABCC1
oxidative stress MRP1 ABCC1
inflammatory responses MRP1 ABCC1
transporter MRP1 ABCC1
multidrug-resistance MRP1 ABCC1
glutathione MRP1 ABCC1
GSH MRP2 ABCC2
vesicular transport MRP1 ABCC1
assay MRP1 ABCC1
nucleotide trapping MRP1 ABCC1
dye transport MRP1 ABCC1
ADME MRP1 ABCC1
Absorption MRP1 ABCC1
Distribution MRP1 ABCC1
Metabolism MRP1 ABCC1
Excretion MRP2 ABCC2
early ADME MRP1 ABCC1
in-vitro system MRP1 ABCC1
drug metabolism MRP1 ABCC1
nucleotide trapping MRP1 ABCC1
dye transport MRP1 ABCC1
efflux transporter MRP1 ABCC1
biovavailability MRP1 ABCC1
xenobiotics MRP1 ABCC1
toxicity MRP1 ABCC1
screening MRP1 ABCC1
cancer drug resistance MRP1 ABCC1
hydrophobic drugs MRP1 ABCC1
penetration MRP1 ABCC1
pharmacological barrier MRP1 ABCC1
drug interaction MRP1 ABCC1
pharmacokinetics MRP1 ABCC1
DMPK MRP1 ABCC1
chemotherapy MRP1 ABCC1
anticancer drug MRP1 ABCC1
resistant tumor cell MRP1 ABCC1
lead optimization MRP1 ABCC1
HTS MRP1 ABCC1
drug development MRP2 ABCC2
pharmacology MRP1 ABCC1
daunorubicin MRP1 ABCC1
aflatoxin B1 MRP1 ABCC1
aflatoxin B1-glutathione conjugate MRP1 ABCC1
benzbromarone MRP1 ABCC1
furosemide MRP1 ABCC1
indomethacin MRP1 ABCC1
LTC4 MRP1 ABCC1
MK571 MRP1 ABCC1
Penicillin G MRP1 ABCC1
rifampicin MRP1 ABCC1
RU 486 MRP1 ABCC1
sulfinpyrazone MRP1 ABCC1
doxorubicin MRP1 ABCC1
clorambucil MRP1 ABCC1
clorambucil-glutathione conjugate MRP1 ABCC1
daunomycin MRP1 ABCC1
daunomycin-glutathione conjugate MRP1 ABCC1
daunorubicin MRP1 ABCC1
daunorubicin-glutathione conjugate MRP1 ABCC1
cyclosporin A MRP1 ABCC1
genistein MRP1 ABCC1
calcein AM MRP1 ABCC1
calcein AM MRP1 ABCC1
membrane MRP2 ABCC2
liver MRP2 ABCC2
bile MRP2 ABCC2
organic anion MRP2 ABCC2
assay MRP2 ABCC2
vesicular transport MRP2 ABCC2
nucleotide trapping MRP2 ABCC2
screening MRP2 ABCC2
Dubin-Johnson MRP2 ABCC2
bilirubin MRP2 ABCC2
efflux transport MRP2 ABCC2
organic anion transport MRP2 ABCC2
ADME MRP2 ABCC2
Distribution MRP2 ABCC2
Metabolism MRP2 ABCC2
Absorption MRP2 ABCC2
Excretion MRP2 ABCC2
early ADME MRP2 ABCC2
in-vitro system MRP2 ABCC2
drug metabolism MRP2 ABCC2
multidrug resistance MRP2 ABCC2
hydrophobic drugs MRP2 ABCC2
penetration MRP2 ABCC2
pharmacological barrier MRP2 ABCC2
hepatobiliary secretion MRP2 ABCC2
kidney secretion MRP2 ABCC2
cancer drug resistance MRP2 ABCC2
drug interaction MRP2 ABCC2
bioavailability MRP2 ABCC2
DMPK MRP2 ABCC2
chemotherapy MRP2 ABCC2
resistant tumor cell MRP2 ABCC2
anticancer drug MRP2 ABCC2
lead optimization MRP2 ABCC2
drug development MRP2 ABCC2
HTS MRP2 ABCC2
pharmacology MRP2 ABCC2
phenylimidazol[4 5-b]pyridine MRP2 ABCC2
somatostatin MRP2 ABCC2
GSH MRP2 ABCC2
PhIP MRP2 ABCC2
somatostatin analogues MRP2 ABCC2
GSH conjugates MRP2 ABCC2
CPT11 MRP2 ABCC2
irinotecan MRP2 ABCC2
endothelin 1 MRP2 ABCC2
estradiol 17-ß-D-glucuronide MRP2 ABCC2
grepafloxacine MRP2 ABCC2
HIV protease inhibitor MRP2 ABCC2
methotrexate MRP2 ABCC2
PAH MRP2 ABCC2
pravastatin MRP2 ABCC2
probenecid MRP2 ABCC2
BSP MRP2 ABCC2
ouabain MRP2 ABCC2
taxol MRP2 ABCC2
telmisaltan MRP2 ABCC2
calcein AM MRP2 ABCC2
furosemide MRP2 ABCC2
Penicillin G MRP2 ABCC2
cefodizime MRP2 ABCC2
cyclosporin A MRP2 ABCC2
genistein MRP2 ABCC2
glibenclamine MRP2 ABCC2
indomethacin MRP2 ABCC2
LTC4 MRP2 ABCC2
MK-571 MRP2 ABCC2
phenobarbital MRP2 ABCC2
quinidine MRP2 ABCC2
rifampicin MRP2 ABCC2
sulfinpyrazone MRP2 ABCC2
sulfinpyrazone MRP2 ABCC2
sulfinpyrazone MRP2 ABCC2 MRP2 ABCC2
drug resistance MRP3 ABCC3
screening MRP3 ABCC3
vesicular transport MRP3 ABCC3
assay MRP3 ABCC3
ADME MRP3 ABCC3
Absorption MRP3 ABCC3
Distribution MRP4 ABCC4
Metabolism MRP5 ABCC5
Excretion MRP6 ABCC6
early ADME MRP3 ABCC3
in-vitro system MRP3 ABCC3
drug metabolism MRP3 ABCC3
drug interaction MRP3 ABCC3
drug development MRP3 ABCC3
organic ion MRP3 ABCC3
efflux transport MRP3 ABCC3
pharmacokinetics MRP3 ABCC3
DMPK MRP3 ABCC3
lead optimization MRP3 ABCC3
HTS MRP3 ABCC3
pharmacology MRP3 ABCC3
glycocholate MRP3 ABCC3
taurocholate MRP3 ABCC3
3H-E217bG MRP3 ABCC3
3H-Methotrexate MRP3 ABCC3
3H-Folic acid MRP3 ABCC3
3H-leucovorin MRP3 ABCC3
furosemid MRP3 ABCC3
benzbromarone MRP3 ABCC3
indomethacine MRP3 ABCC3
E217bG MRP3 ABCC3
E217bG MRP3 ABCC3
E217bG MRP3 ABCC3
E217bG MRP3 ABCC3 MRP4 ABCC4
membrane MRP4 ABCC4
assay MRP4 ABCC4
screening MRP4 ABCC4
nucleotide analogue transport MRP4 ABCC4
ADME MRP4 ABCC4
Absorption MRP4 ABCC4
Distribution MRP5 ABCC5
Metabolism MRP6 ABCC6
Excretion MRP7 ABCC7
early ADME MRP4 ABCC4
in-vitro system MRP4 ABCC4
drug metabolism MRP4 ABCC4
pharmacology MRP4 ABCC4
3H-E217bG MRP4 ABCC4
3H-Methotrexate MRP4 ABCC4
3H-Folic acid MRP4 ABCC4
3H-Leucovorin MRP4 ABCC4
3H-DHEAS MRP4 ABCC4
cGMP MRP4 ABCC4
cAMP MRP4 ABCC4
Methotrexate MRP4 ABCC4
Zaprinast MRP4 ABCC4
E217bG MRP4 ABCC4
DHEAS MRP4 ABCC4
Sulfinpyrazone MRP4 ABCC4
MK-571 MRP4 ABCC4
Probenecid MRP4 ABCC4
Probenecid MRP4 ABCC4
pharmacology MRP5 ABCC5
nucleoside transport MRP5 ABCC5
3H-cAMP MRP5 ABCC5
3H-6-SH-purine MRP5 ABCC5
3H-cGMP MRP5 ABCC5
3H-alaninyl-d4TMP MRP5 ABCC5
Zaprinast MRP5 ABCC5
Benzbromarone MRP5 ABCC5
MK-571 MRP5 ABCC5
Sulfinpyrazone MRP5 ABCC5
Probenecid MRP5 ABCC5
cGMP MRP5 ABCC5
cAMP MRP5 ABCC5
cAMP MRP5 ABCC5
cAMP MRP5 ABCC5 MRP6 ABCC6
cAMP MRP5 ABCC5 MRP6 ABCC6 MRP6 ABCC6
cAMP MRP5 ABCC5 MRP6 ABCC6 MRP6 ABCC6 MRP6 ABCC6
cAMP MRP5 ABCC5 MRP6 ABCC6 MRP6 ABCC6 MRP6 ABCC6 MRP6 ABCC6
cAMP MRP5 ABCC5 MRP6 ABCC6 MRP6 ABCC6 MRP6 ABCC6 MRP6 ABCC6 MRP6 ABCC6
cAMP MRP5 ABCC5 MRP6 ABCC6 MRP6 ABCC6 MRP6 ABCC6 MRP6 ABCC6 MRP6 ABCC6 MRP6 ABCC6
cAMP MRP5 ABCC5 MRP6 ABCC6 MRP6 ABCC6 MRP6 ABCC6 MRP6 ABCC6 MRP6 ABCC6 MRP6 ABCC6
cAMP MRP5 ABCC5 MRP6 ABCC6 MRP6 ABCC6 MRP6 ABCC6 MRP6 ABCC6 MRP6 ABCC6 MRP6 ABCC6 MXR ABCG2
lead optimization MXR ABCG2
HTS MXR ABCG2
drug development MXR ABCG2
membrane MXR ABCG2
cancer drug resistance MXR ABCG2
screening MXR ABCG2
vesicular transport MXR ABCG2
nucleotide trapping MXR ABCG2
assay MXR ABCG2
pharmacokinetics MXR ABCG2
pharmacological barrier MXR ABCG2
dye transport MXR ABCG2
ADME MXR ABCG2
Absorption MXR ABCG2
Distribution MXR ABCG2
Metabolism MXR ABCG2
excretion MXR ABCG2
early ADME MXR ABCG2
in-vitro system MXR ABCG2
drug metabolism MXR ABCG2
drug interaction MXR ABCG2
efflux transport MXR ABCG2
xenobiotics MXR ABCG2
DMPK MXR ABCG2
chemotherapy MXR ABCG2
anticancer drugs MXR ABCG2
resistant tumor cells MXR ABCG2
pharmacology MXR ABCG2
topotecan MXR ABCG2
mitoxantrone MXR ABCG2
irinotecan MXR ABCG2
SN-38 MXR ABCG3
9-amino campto MXR ABCG2
indolocarbazoles MXR ABCG2
NB506 MXR ABCG2
J-107088 MXR ABCG2
Topo 1 inhibitors MXR ABCG2
methotrexate MXR ABCG2
anthracyclines MXR ABCG2
Dox MXR ABCG2
DNR MXR ABCG2
IDA MXR ABCG2
flavopiridol MXR ABCG2
quinazolines MXR ABCG2
HER tyrosine kinase inhibitor MXR ABCG2
prazosine MXR ABCG2
CI1033 MXR ABCG2
fumitremorgin C MXR ABCG2
FTC MXR ABCG2
GF120918 MXR ABCG2
prazocine MXR ABCG2
iressa MXR ABCG2
BIB-E MXR ABCG2
novobiocin MXR ABCG2
VX-710 MXR ABCG2
VX853 MXR ABCG2
estrogens MXR ABCG2
tamoxifene MXR ABCG2
tamoxifene MXR ABCG2
membrane Bsep Abcb11
FXR Bsep Abcb11
bile salt Bsep Abcb11
intrahepatic cholestasis Bsep Abcb11
intrahepatic cholestasis Bsep Abcb11 Bsep Abcb11
efflux transport Bsep Abcb11
cancer drug resistance Bsep Abcb11
screening Bsep Abcb11
vesicular transport Bsep Abcb11
drug interaction Bsep Abcb11
assay Bsep Abcb11
pharmacokinetics Bsep Abcb11
ADME Bsep Abcb11
Absorption Bsep Abcb11
Distribution Bsep Abcb11
Metabolism Bsep Abcb11
Excretion Bsep Abcb11
early ADME Bsep Abcb11
in-vitro system Bsep Abcb11
drug metabolism Bsep Abcb11
pharmacology Bsep Abcb11
bosentan Bsep Abcb11
troglitazone Bsep Abcb11
3H-Taurocholate Bsep Abcb11
3H-Glycocholate Bsep Abcb11
3H-Taurochenodesoxycholate Bsep Abcb11
3H-Tauroursodesoxycholate Bsep Abcb11
Taurochenodesoxycholate Bsep Abcb11
Glibenclamide Bsep Abcb11
Taurocholate Bsep Abcb11
Glycocholate Bsep Abcb11
Rifamicin SV Bsep Abcb11
Rifampicin Bsep Abcb11
Cyclosporin A Bsep Abcb11
Rifamicin SV Bsep Abcb11
Glibenclamide Bsep Abcb11
Glibenclamide Bsep Abcb11
liver ABCB4 MDR3
membrane ABCB4 MDR3
lead optimization ABCB4 MDR3
HTS ABCB4 MDR3
pharmacology ABCB4 MDR3
drug development ABCB4 MDR3
fatty acid secretion ABCB4 MDR3
modulators ABCB4 MDR3
environmental toxicity ABCB4 MDR3
ADME ABCB4 MDR3
Absorption ABCB4 MDR3
Distribution ABCB5 MDR4
Metabolism ABCB6 MDR5
Excretion ABCB7 MDR6
early ADME ABCB4 MDR3
in-vitro system ABCB4 MDR3
drug metabolism ABCB4 MDR3
nucleotide trapping ABCB4 MDR3
assay ABCB4 MDR3
phosphatidyl-choline transport ABCB4 MDR3
phosphatidyl-choline transport ABCB4 MDR3
3H-Methyl-quinidine rMdr1b Rat Mdr1b
3H-Methyl-quinine rMdr1b Rat Mdr1b
Verapamil rMdr1b Rat Mdr1b
Quinidine rMdr1b Rat Mdr1b
Erithromycin rMdr1b Rat Mdr1b
Prazosin rMdr1b Rat Mdr1b
Ritonavir rMdr1b Rat Mdr1b
Digoxin rMdr1b Rat Mdr1b
Doxorubicin rMdr1b Rat Mdr1b
Methotrexate rMdr1b Rat Mdr1b
Ranitidine rMdr1b Rat Mdr1b
Ranitidine rMdr1b Rat Mdr1b
3H-E217bG rMrp2 Rat Mrp2
3H-LTC4 rMrp2 Rat Mrp2
3H-Methotrexate rMrp2 Rat Mrp2
3H-BQ123 rMrp2 Rat Mrp2
NEM-GS rMrp2 Rat Mrp2
Probenecid rMrp2 Rat Mrp2
Sulfinpyrazone rMrp2 Rat Mrp2
Indomethacin rMrp2 Rat Mrp2
Methotrexate rMrp2 Rat Mrp2
Furosemid rMrp2 Rat Mrp2
Benzbromarone rMrp2 Rat Mrp2
Benzbromarone rMrp2 Rat Mrp2
MultiDrugQuantTM assay kit MDQkit
haematology MultiDrugQuant
solid tumor MultiDrugQuant clinical trial
leukemia MultiDrugQuant
leukemia MultiDrugQuant MultiDrugQuant
leukemia MultiDrugQuant MultiDrugQuant
absorption ABC transporter
ADME ABC transporter
xenobiotics ABC transporter
screening ABC transporter
vesicular transport ABC transporter
membrane ABC transporter
membrane assay ABC transporter
bioaccumulation ABC transporter
multispecificity ABC transporter
drug-drug interaction ABC transporter
drug-drug interaction multispecificity
calcein assay ABC transporter
ATPase assay ABC transporter
efflux transport ABC transporter
modulation ABC transporter
multidrug resistance ABC transporter
CSF penetration ABC transporter
DMPK ABC transporter
rapid filtration ABC transporter
nucleotide trapping ABC transporter
Sf 9 cells ABC transporter
vesicular transport assay ABC transporter
monolayer efflux assay ABC transporter
vanadate dependent nucleotide trapping ABC transporter

 

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Last updated: May 15, 2008
This page contains information about following topics: Pgp, P-gp, MDR1, ABCB1, P-glycoprotein, MRP1, ABCC2, MRP2, ABCC2, cMOAT, MRP3, ABCC3, cMOAT-2, MRP4, ABCC4, MOATB, MRP5, ABCC6, BCRP, MXR, ABCG2, BSEP, ABCB11, ratBsep, mouse bsep, mouse bcrp, mouse mxr, rat Mdr, rat Mrp2, MDR3, NTCP, SLC10A1, rat Ntcp, OATP1B1, OATP-C, OATP2, SLCO1B1, OATP1B3, OATP8, SLCO1B3, OATP2B1, OATP-B, SLCO2B1, rat Oatp1a1, Oatp1, rat Oatp1a4, Oatp2, rat Oatp1b2, Oatp4, PEPT1, SLC15A1, PEPT2, SLC15B2membrane transporter,calcein assay kit,screening,MDR1,MRP1,MRP2,MRP3,MRP4,MXR,BSEP,blood-brain barrier, cMOAT-3, MRP5, ABCC5, cMOAT-4, MRP6, ABCC6.