Vesicular Transport Membranes

Product Cell Line Transporter Technology Membrane Type Probe Substrate Readout Reference Inhibitor Positive Control Dynamic Range Shipping Option
SB BCRP HEK293 Membrane BCRP
Vesicular Transport Assay
HEK293 E3S >7 From EU and US
SB BSEP HEK293 Membrane BSEP
Vesicular Transport Assay
HEK293 Taurocholate >15 From EU and US
SB MDR1/P-gp HEK293 Membrane MDR1/P-gp
Vesicular Transport Assay
HEK293 NMQ >5 From EU and US
SB MRP1 HEK293 Membrane MRP1
Vesicular Transport Assay
HEK293 E217ßG >3 From EU and US
SB MRP2 HEK293 Membrane MRP2
Vesicular Transport Assay
HEK293 E217ßG >10 From EU and US
SB MRP3 HEK293 Membrane MRP3
Vesicular Transport Assay
HEK293 E217ßG >10 From EU and US
SB MRP4 HEK293 Membrane MRP4
Vesicular Transport Assay
HEK293 DHEAS >5 From EU and US
SB MRP5 HEK293 Membrane MRP5
Vesicular Transport Assay
HEK293 CDCF >3 From EU and US
SB cyMdr1 HEK293 Membrane Mdr1 - cynomolgus monkey
Vesicular Transport Assay
HEK293 NMQ >5 From EU and US
SB cyBcrp HEK293 Membrane Bcrp - cynomolgus monkey
Vesicular Transport Assay
HEK293 E3S >5 From EU and US
SB cyBsep HEK293 Membrane Bsep - cynomolgus monkey
Vesicular Transport Assay
HEK293 Taurocholate >5 From EU and US
SB dogBsep HEK293 Membrane Bsep - dog
Vesicular Transport Assay
HEK293 Taurocholate >10 From EU and US
SB mouseBcrp HEK293 Membrane Bcrp - mouse
Vesicular Transport Assay
HEK293 E3S >2 From EU
SB mouseMdr1a HEK293 Membrane Mdr1a - mouse
Vesicular Transport Assay
HEK293 NMQ >5 From EU
SB ratBcrp HEK293 Membrane Bcrp - rat
Vesicular Transport Assay
HEK293 Estrone-3-sulfate >3 From EU
SB ratBsep HEK293 Membrane Bsep - rat
Vesicular Transport Assay
HEK293 Taurocholate >5 From EU and US
SB ratMdr1b Sf9 HAM Membrane Mdr1b - rat
Vesicular Transport Assay
Sf9-HAM NMQ >4 From EU
SB ratMrp2 HEK293 Membrane Mrp2 - rat
Vesicular Transport Assay
HEK293 E217ßG >5 From EU and US
SB ratMrp3 HEK293 Membrane Mrp3 - rat
Vesicular Transport Assay
HEK293 E217ßG >5 From EU and US
SB BSEP Hi5 Membrane BSEP
Vesicular Transport Assay
Hi5 Taurocholate >5 From EU

Description

Membrane Preparations for Vesicular Transport Assays (VT) are suitable for general drug-efflux transporter interaction studies. Both substrate and inhibitor interactions can be assessed using vesicles. The success of substrate interaction studies strongly depends on the passive permeability of the compound. High permeability substrates might not be detected. Control Membranes with no-, or significantly lower transporter activity are also available. For the scientific background of our vesicular transport assays, please click here.

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