| Service |
Cell Line |
Transporter |
Technology |
Membrane Type |
Probe Substrate |
Read Out |
Reference Inhibitor |
Positive Control |
Dynamic Range |
| Asbt-rat Uptake Transporter Assay |
|
Asbt - rat
|
Uptake Transporter Assay
|
|
Taurocholate |
|
Taurochenodeoxycholate (TCDC) |
|
|
| ASBT Uptake Transporter Assay |
|
ASBT
|
Uptake Transporter Assay
|
|
Taurocholate |
|
Taurochenodeoxycholate (TCDC) |
|
|
| ASCT1 Uptake Transporter Assay- Serine |
|
ASCT1
|
Uptake Transporter Assay
|
|
Serine |
|
L-cysteine |
|
|
| ASCT2 Uptake Transporter Assay- Serine |
|
ASCT2
|
|
|
Serine |
|
L-cysteine |
|
|
| CNT1 Uptake Transporter Assay |
|
CNT1
|
Uptake Transporter Assay
|
|
Uridine |
|
Adenosine |
|
|
| CNT2 Uptake Transporter Assay |
|
CNT2
|
Uptake Transporter Assay
|
|
Uridine |
|
Adenosine |
|
|
| CNT3 Uptake Transporter Assay |
|
CNT3
|
Uptake Transporter Assay
|
|
Uridine |
|
2′-Deoxycytidine |
|
|
| Ent1-Rat Uptake Transporter Assay |
|
Ent1-rat
|
Uptake Transporter Assay
|
|
Adenosine |
|
NBMPR (0.01 µM) |
|
|
| ENT1 Uptake Transporter Assay |
|
ENT1
|
Uptake Transporter Assay
|
|
Uridine |
|
Dilazep |
|
|
| ENT2 Uptake Transporter Assay |
|
ENT2
|
Uptake Transporter Assay
|
|
Adenosine |
|
Dipyridamole |
|
|
| ENT4 Uptake Transporter Assay |
|
ENT4
|
Uptake Transporter Assay
|
|
MPP+ |
|
Pyrimethamine |
|
|
| HPT1 Uptake Transporter Assay |
|
HPT1
|
Uptake Transporter Assay
|
|
Gly-Sar |
|
Cefadroxil |
|
|
| LAT1 Uptake Transporter Assay |
|
LAT1
|
Uptake Transporter Assay
|
|
Leucine |
|
JPH203 |
|
|
| LAT2 Uptake Transporter Assay |
|
LAT2
|
Uptake Transporter Assay
|
|
Leucine |
|
JX009 |
|
|
| MATE1 Uptake Transporter Assay - Metformin |
|
MATE1
|
Uptake Transporter Assay
|
|
Metformin |
|
Pyrimethamine |
|
|
| MATE1 Uptake Transporter Assay - Tetraethylammonium chloride (TEA) |
|
MATE1
|
Uptake Transporter Assay
|
|
Tetraethylammonium chloride (TEA) |
|
Pyrimethamine |
|
|
| MATE2-K Uptake Transporter Assay - Metformin |
|
MATE2
|
Uptake Transporter Assay
|
|
Metformin |
|
Pyrimethamine |
|
|
| MATE2-K Uptake Transporter Assay - Tetraethylammonium chloride (TEA) |
|
MATE2
|
Uptake Transporter Assay
|
|
Tetraethylammonium chloride (TEA) |
|
Pyrimethamine |
|
|
| MCT10 Uptake Transporter Assay |
|
MCT10
|
Uptake Transporter Assay
|
|
Triiodothyronine (T3) |
|
Imatinib mesylate |
|
|
| MCT8 Uptake Transporter Assay |
|
MCT8
|
Uptake Transporter Assay
|
|
Triiodothyronine (T3) |
|
Sorafenib |
|
|
| Nis - Rat Uptake Transporter Assay |
|
Nis - rat
|
Uptake Transporter Assay
|
|
Iodide |
|
Potassium perchlorate |
|
|
| NIS Uptake Transporter Assay |
|
NIS
|
Uptake Transporter Assay
|
|
Iodide |
|
Potassium perchlorate |
|
|
| Ntcp- Cynomolgus monkey Uptake Transporter Assay |
|
Ntcp - cynomolgus monkey
|
Uptake Transporter Assay
|
|
Taurocholate |
|
Taurochenodeoxycholate (TCDC) |
|
|
| Ntcp- Rat Uptake Transporter Assay |
|
Ntcp - rat
|
Uptake Transporter Assay
|
|
Taurocholate |
|
Troglitazone |
|
|
| NTCP Uptake Transporter Assay |
|
NTCP
|
Uptake Transporter Assay
|
|
Taurocholate |
|
Taurochenodeoxycholate (TCDC) |
|
|
| Oat1- Rat Uptake Transporter Assay |
|
Oat1 - rat
|
Uptake Transporter Assay
|
|
p-Aminohippuric acid (PAH) |
|
Benzbromarone |
|
|
| OAT1 Uptake Transporter Assay - Para-Aminohippuric acid (PAH) |
|
OAT1
|
Uptake Transporter Assay
|
|
p-Aminohippuric acid (PAH) |
|
Benzbromarone |
|
|
| OAT1 Uptake Transporter Assay - Tenofovir |
|
OAT1
|
Uptake Transporter Assay
|
|
Tenofovir |
|
Probenecid |
|
|
| OAT1 Uptake Transporter Assay - Uric acid |
|
OAT1
|
Uptake Transporter Assay
|
|
Uric acid |
|
Benzbromarone |
|
|
| OAT2v1 Uptake Transporter Assay - cGMP |
|
OAT2
|
Uptake Transporter Assay
|
|
cGMP |
|
Indomethacin |
|
|
| OAT2v1 Uptake Transporter Assay - Creatinine |
|
OAT2
|
Uptake Transporter Assay
|
|
Creatinine |
|
Indomethacin |
|
|
| OAT2v1 Uptake Transporter Assay - Uric acid |
|
OAT2
|
Uptake Transporter Assay
|
|
Uric acid |
|
Indomethacin |
|
|
| OAT3 Uptake Transporter Assay - Estrone 3-sulfate (E3S) |
|
OAT3
|
Uptake Transporter Assay
|
|
Estrone-3-Sulfate (E3S) |
|
Probenecid |
|
|
| OAT3 Uptake Transporter Assay - Methotrexate (MTX) |
|
OAT3
|
Uptake Transporter Assay
|
|
Methotrexate (MTX) |
|
Probenecid |
|
|
| OAT3 Uptake Transporter Assay - Uric acid |
|
OAT3
|
Uptake Transporter Assay
|
|
Uric acid |
|
Benzbromarone |
|
|
| OAT4 Uptake Transporter Assay- Estrone-3-sulfate |
|
OAT4
|
Uptake Transporter Assay
|
|
Estrone-3-sulfate |
|
Benzbromarone |
|
|
| OAT4 Uptake Transporter Assay- Uric acid |
|
OAT4
|
Uptake Transporter Assay
|
|
Uric acid |
|
Benzbromarone |
|
|
| OAT7 Uptake Transporter Assay |
|
OAT7
|
Uptake Transporter Assay
|
|
Estrone-3-Sulfate (E3S) |
|
Sulfobromophthalein |
|
|
| Oatp1a1 - Rat Uptake Transporter Assay - Estrone 3-sulfate (E3S) |
|
Oatp1a1 - rat
|
Uptake Transporter Assay
|
|
Estrone-3-Sulfate (E3S) |
|
Dehydroisoandrosterone 3-sulfate |
|
|
| Oatp1a1 - Rat Uptake Transporter Assay - Taurocholate |
|
Oatp1a1 - rat
|
Uptake Transporter Assay
|
|
Taurocholate |
|
Dehydroisoandrosterone 3-sulfate |
|
|
| OATP1A2 Uptake Transporter Assay |
|
OATP1A2
|
Uptake Transporter Assay
|
|
Estrone-3-Sulfate (E3S) |
|
Sulfobromophthalein (BSP) |
|
|
| Oatp1a4 - Rat Uptake Transporter Assay |
|
Oatp1a4 - rat
|
Uptake Transporter Assay
|
|
Taurocholate |
|
Rifampicin |
|
|
| Oatp1b1- Cynomolgus monkey Uptake Transporter Assay - Estrone 3-sulfate (E3S) |
|
Oatp1b1 - cynomolgus monkey
|
Uptake Transporter Assay
|
|
Estrone 3-sulfate (E3S) |
|
Fluvastatin |
|
|
| Oatp1b1 - Cynomolgus monkey Uptake Transporter Assay - β-Estradiol 17-(β-D-glucuronide) |
|
Oatp1b1 - cynomolgus monkey
|
Uptake Transporter Assay
|
|
β-Estradiol 17-(β-D-glucuronide) |
|
Rifampicin |
|
|
| OATP1B1 Uptake Transporter Assay - Estrone 3-sulfate (E3S) |
|
OATP1B1
|
Uptake Transporter Assay
|
|
Estrone-3-Sulfate (E3S) |
|
Cyclosporin A |
|
|
| OATP1B1 Uptake Transporter Assay - Coproporphyrin I |
|
OATP1B1
|
Uptake Transporter Assay
|
|
Coproporphyrin I |
|
Rifampicin |
|
|
| OATP1B1 Uptake Transporter Assay - β-Estradiol 17-(β-D-glucuronide) |
|
OATP1B1
|
Uptake Transporter Assay
|
|
β-Estradiol 17-(β-D-glucuronide) |
|
Rifampicin |
|
|
| OATP1B1 Uptake Transporter Assay - Olmesartan |
|
OATP1B1
|
Uptake Transporter Assay
|
|
Olmesartan |
|
Rifampicin |
|
|
| OATP1B1 Uptake Transporter Assay - Rosuvastatin |
|
OATP1B1
|
Uptake Transporter Assay
|
|
Rosuvastatin |
|
Rifampicin |
|
|
| Oatp1b2- Rat Uptake Transporter Assay |
|
Oatp1b2 - rat
|
Uptake Transporter Assay
|
|
Taurocholate |
|
Taurochenodeoxycholate (TCDC) |
|
|
| Oatp1b3- Cynomolgus monkey Uptake Transporter Assay - β-Estradiol 17-(β-D-glucuronide) |
|
Oatp1b3 -cynomolgus monkey
|
Uptake Transporter Assay
|
|
β-Estradiol 17-(β-D-glucuronide) |
|
Cyclosporin A |
|
|
| Oatp1b3- Cynomolgus monkey Uptake Transporter Assay - CCK8 |
|
Oatp1b3 -cynomolgus monkey
|
Uptake Transporter Assay
|
|
CCK8 |
|
Cyclosporin A |
|
|
| OATP1B3 Uptake Transporter Assay - CCK8 |
|
OATP1B3
|
Uptake Transporter Assay
|
|
CCK8 |
|
Rifampicin |
|
|
| OATP1B3 Uptake Transporter Assay - Coproporphyrin I |
|
OATP1B3
|
Uptake Transporter Assay
|
|
Coproporphyrin I |
|
Rifampicin |
|
|
| OATP1B3 Uptake Transporter Assay - Coproporphyrin III |
|
OATP1B3
|
Uptake Transporter Assay
|
|
Coproporphyrin III |
|
Rifampicin |
|
|
| OATP1B3 Uptake Transporter Assay - Fluo-3 |
|
OATP1B3
|
Uptake Transporter Assay
|
|
Fluo-3 |
|
Fluvastatin |
|
|
| OATP1B3 Uptake Transporter Assay - Olmesartan |
|
OATP1B3
|
Uptake Transporter Assay
|
|
Olmesartan |
|
Rifampicin |
|
|
| OATP1B3 Uptake Transporter Assay - Rosuvastatin |
|
OATP1B3
|
Uptake Transporter Assay
|
|
Rosuvastatin |
|
Cyclosporin A |
|
|
| OATP1B3 Uptake Transporter Assay - β-Estradiol 17-(β-D-glucuronide) |
|
OATP1B3
|
Uptake Transporter Assay
|
|
β-Estradiol 17-(β-D-glucuronide) |
|
Rifampicin |
|
|
| OATP2A1 Uptake Transporter Assay |
|
OATP2A1
|
Uptake Transporter Assay
|
|
Prostaglandin-E2 |
|
Diclofenac |
|
|
| Oatp2b1- Cynomolgus monkey Uptake Transporter Assay |
|
Oatp2b1 - cynomolgus monkey
|
Uptake Transporter Assay
|
|
Estrone 3-sulfate (E3S) |
|
Sulfasalazine |
|
|
| OATP2B1 Uptake Transporter Assay - Estrone 3-sulfate (E3S) |
|
OATP2B1
|
Uptake Transporter Assay
|
|
Estrone-3-Sulfate (E3S) |
|
Rifamycin SV |
|
|
| OATP2B1 Uptake Transporter Assay - Coproporphyrin III |
|
OATP2B1
|
Uptake Transporter Assay
|
|
Coproporphyrin III |
|
Erlotinib |
|
|
| OATP2B1 Uptake Transporter Assay - Rosuvastatin |
|
OATP2B1
|
Uptake Transporter Assay
|
|
Rosuvastatin |
|
Erlotinib |
|
|
| OCT1 Uptake Transporter Assay - Metformin |
|
OCT1
|
Uptake Transporter Assay
|
|
Metformin |
|
Verapamil |
|
|
| OCT1 Uptake Transporter Assay - Sumatriptan |
|
OCT1
|
Uptake Transporter Assay
|
|
Sumatriptan |
|
Verapamil |
|
|
| OCT1 Uptake Transporter Assay - Tetraethylammonium chloride (TEA) |
|
OCT1
|
Uptake Transporter Assay
|
|
Tetraethylammonium chloride (TEA) |
|
Verapamil |
|
|
| OCT2 Uptake Transporter Assay - Metformin |
|
OCT2
|
Uptake Transporter Assay
|
|
Metformin |
|
Clonidine |
|
|
| OCT2 Uptake Transporter Assay - Creatinine |
|
OCT2
|
Uptake Transporter Assay
|
|
Creatinine |
|
Verapamil |
|
|
| OCT2 Uptake Transporter Assay - MPP+ |
|
OCT2
|
Uptake Transporter Assay
|
|
MPP+ |
|
Phenoxybenzamine |
|
|
| OCT2 Uptake Transporter Assay - Tetraethylammonium chloride (TEA) |
|
OCT2
|
Uptake Transporter Assay
|
|
Tetraethylammonium chloride (TEA) |
|
Verapamil |
|
|
| OCT3 Uptake Transporter Assay |
|
OCT3
|
Uptake Transporter Assay
|
|
MPP+ |
|
Quinidine |
|
|
| OCTN1 Uptake Transporter Assay |
|
OCTN1
|
Uptake Transporter Assay
|
|
Tetraethylammonium-chloride (TEA) |
|
Verapamil |
|
|
| Octn2- Rat Uptake Transporter Assay |
|
Octn2 - rat
|
Uptake Transporter Assay
|
|
Carnitine |
|
Verapamil |
|
|
| OCTN2 Uptake Transporter Assay |
|
OCTN2
|
Uptake Transporter Assay
|
|
Carnitine |
|
Verapamil |
|
|
| OSTα/β- Rat Uptake Transporter Assay |
|
Ost α and β - rat
|
Uptake Transporter Assay
|
|
Estrone 3-sulfate (E3S) |
|
Ko143 |
|
|
| OSTα/β Uptake Transporter Assay |
|
OST α and β
|
Uptake Transporter Assay
|
|
Estrone 3-sulfate (E3S) |
|
Ko143 |
|
|
| PEPT1 Uptake Transporter Assay |
|
PEPT1
|
Uptake Transporter Assay
|
|
Gly-Sar |
|
Tyr-Phe |
|
|
| PEPT2 Uptake Transporter Assay |
|
PEPT2
|
Uptake Transporter Assay
|
|
Gly-Sar |
|
Cefadroxil |
|
|
| RFVT3 Uptake Transporter Assay - Riboflavin |
|
RFVT3
|
Uptake Transporter Assay
|
|
Riboflavin |
|
FMN (1,000 µM) |
|
|
| SGLT1 Uptake Transporter Assay |
|
SGLT1
|
Uptake Transporter Assay
|
|
methyl-α-D-glucopyranoside |
|
Phloridzin |
|
|
| Sglt2-dog Uptake Transporter Assay |
|
Sglt2 - dog
|
Uptake Transporter Assay
|
|
Methyl-α-D-glucopyranoside |
|
Dapagliflozin |
|
|
| Sglt2-mouse Uptake Transporter Assay |
|
Sglt2 - mouse
|
Uptake Transporter Assay
|
|
Methyl-α-D-glucopyranoside |
|
Dapagliflozin |
|
|
| SGLT2 Uptake Transporter Assay |
|
SGLT2
|
Uptake Transporter Assay
|
|
Methyl-α-D-glucopyranoside |
|
Dapagliflozin |
|
|
| SGLT5 Uptake Transporter Assay |
|
SGLT5
|
Uptake Transporter Assay
|
|
Fructose |
|
Dapagliflozin |
|
|
| SGLT6 Uptake Transporter Assay |
|
SGLT6
|
Uptake Transporter Assay
|
|
Myo-Inositol |
|
Dapagliflozin |
|
|
| THTR1 Uptake Transporter Assay |
|
THTR1
|
Uptake Transporter Assay
|
|
Thiamine |
|
Amprolium |
|
|
| THTR2 Uptake Transporter Assay |
|
THTR2
|
Uptake Transporter Assay
|
|
Thiamine |
|
Fedratinib |
|
|
| URAT1 Uptake Transporter Assay - Orotic acid |
|
URAT1
|
Uptake Transporter Assay
|
|
Orotic acid |
|
Benzbromarone |
|
|
| URAT1 Uptake Transporter Assay - Uric acid |
|
URAT1
|
Uptake Transporter Assay
|
|
Uric acid |
|
Benzbromarone |
|
|
